Apriso.
375 mg ER
Site of action: colon
Asacol(HD)
Generic mesalamine
800 mg delayed release DR
Site of action: distal ileum- colon
Delzicol
DR mesalamine
Distal ileum- colon
400 mg delayed release
Lialda
DR mesalamine
(Distal ileum - colon)
1.2 g delayed release
Pentasa
Controlled release
Duodenum, jejeunem, ileum, colon
250 mg and 500 mg CR
Canasa.
Suppository mesalamine
Rectum
1000 mg suppository
Rowasa.
Mesalamine enema
4 g (60 ml) enema
Sigmoid colon - rectum
Sulfasalazine
5-Asa I: Ir 1 g PO/ 4x/day DR: 2 g PO 2x/day -\_\_\_\_\_\_\_\_\_\_\_\_\_\_\_\_\_\_ M: it was g PO 2x/day DR: 2 g PO daily
Balsalazide
5-Asa
I: 2.25-3.3 g PO 2x-3x/day
M: 3-6 g PO daily divided conveniently
Olsalazine
5-Asa
I: 750-1500 mg PO 2 x/day
M: 500 mg PO 2x/day