Receptors
Nalmefene
Agonist for Mu, K (Kappa)
Doses
Nalmefene
IV: 15 - 25mcg q2 - 5min
OR
IV: 1 mcg/kg
E 1/2 Time
Nalmefene
10.8 hrs
Metabolism
Nalmefene
Hepatic: Glucuronic acid conjugation
Potency
Nalmefene
Equally potent to naloxone
Side Effects
Nalmefene
Acute pulmonary edema