Esmolol
Mechanism of Action
β1 adrenergic receptor blocker with little to no effect on β2 receptors except at high doses
Esmolol
Class
Beta-blocker, β1 selective
Esmolol
Induction Dose: None
None
Esmolol
Bolus Dose
0.5 mg/kg
Esmolol
Gtt rate
50-300 mcg/kg/min
Esmolol
Common Side Effects / Contraindications
Hypotension
Esmolol
Onset
2 min
Esmolol
Peak
5 min
Esmolol
Distribution half-life (t1/2α)
9-10 min
Esmolol
Metabolism
RBC esterases
Esmolol
Elimination half-life (t1/2 β)/ Active metabolites
9 min